Ola kinoHoomakaukau

Analogs "Ksarelto": uku, olelo ao no ka hoʻohana

Kekahi o na ai ', a e pili ana i ka pharmacological pūʻulu o anticoagulant Luna, i ka lāʻau' o "Ksarelto". Kēia lāʻau inhibits ololi Xa, a me ka ia, ma ka huli, o ka ke keʻena o ka prothrombin activator a me kekahi o na eiiiiiaiou hoʻolako '' eleu koko coagulation (i na waiwai a me analogues "Ksarelto").

I kēia lā lawe mai ho'āʻo nui futile e haalele i ka lāʻau, a e i ka like me keia, a pela no i ka palena iki o kaʻaoʻao loa. Ma hope mau manawa-e hoopau ana ke kākoʻo 'ana i ka pono counterpart - ka lāʻau "Pradaksa". Ke k - wale ae pani i hoopau ai i hiki ke hoʻohana kahi o "Ksarelto" hoʻomākaukau. Kona ano e kokoke'ālike i ka luna, ka mea wale nō likeʻole - kaʻeleu 'Oponopono maʻiʻo, i loko o nā hoomakaukau mea rivaroxaban.

pharmacodynamics

All analogues "Ksarelto" i ka like hopena. Ka mea wale nō ka mea, OAOOUIEeE - ka laupaʻi, a qualitative anakahi o kaʻaoʻao loa. Ka mea wale nō e pono ai mea like o ka lāʻau, i ka mea i like ia i ka mea, o ka lāʻau "Pradaksa".

Kēia lāʻau a me kona Lūkini like paha o ka "Ksarelto" i kauoha nui e wae ai 'i inhibit i ka hana o ololi Xa, oa inhibit ia. Kēia lāʻau i ke kiʻekiʻe ku una bioavailability, naʻe enteral ala hele o ka hooponopono mea Central ia ia.

Central kūlana ma ka cascade o coagulation ololi X ho'ā hope Radio he hope biotransformation ololi Xa Via na, a mawaho coagulation alanui.

hoike

Nō kāu, analogs "Ksarelto" a ua hoʻohana 'ia o ka wa hoomakaukau ia ia iho i loko o ka kēia mau wahi, i hiki:

  • Kāohiʻana a me prophylaxis o ka hahau ana.
  • Kāohiʻana a me ke ola o systemic embolism.

    (Ma na hihia a pau, i ka medicament ua hōʻike ma nā mea maʻi me ka atrial fibrillation, i mea 'ole-valvular kumu.)
  • Removal a Kāohiʻana o plugging o ka hohonu aa koko thrombi.
  • Kāohiʻana o ka recurrence o pulmonary embolism.

Uluwehi O "Pradaksa", i mea like, ua kekahi hōʻike no ka Kāohiʻana o venous thromboembolic hanana i loko o nā mea maʻi i i undergoneʻoki kino e puku i kekahi o na ami o ka lalo lala.

Contraindications

Kekahi Lūkini like paha "Ksarelto" i ka kēia mau contraindications (ka mea hiki e kekahi, akā, wale i ka meaʻuʻuku loa):

  • pā lonoaʻili paha kamepiula hoikeana o allergic reactions i ka waiwai i loaʻa ma loko o ka medicament;
  • ʻeleu kahe ana ke koko a i koʻikoʻi informativeness ma ka lapaʻau ninaninau (e laʻa me, intracavitary kahe ana ke koko a hemorrhage i loko o ka lolo);

  • i kekahi kahua ma a he mea ka māhuahua pilikia o ke kahe ana ke koko ka leo, e laʻa me, ma kaʻeleu ulcer keʻano o ka hanaʻana i loko o ka gastrointestinal'āpana;
  • lāʻau Inc konohiki i loaa like waiwai - pale coagulation;
  • ka hoʻohana 'ana unfractionated heparin ma ka mahele lāʻau pono no kupono ana o ka catheter;
  • likeʻole akepaa maʻi, i ka ulu ana o ka a hiki i kahe ana ke koko mai o kekahi mau etiology;
  • na mea a pau counterparts "Ksarelto" e contraindicated i loko o nā mea maʻi me kaʻaʻa puʻuwai insufficiency, 'ia i loko o kekahi pae;
  • lactose intolerance, lawa ka maʻiʻo o ka galactose i loko o ke kino;
  • hāpai keiki, a lactation;
  • pū ma luna o ka lāʻau a me nā analogs "Ksarelto" he mea he mau makahiki kali 18+.

Mahele o ka poe i lawe i kēia k me ka mālama nui, a ma lalo o ka hooponopono ana o ka hoʻomalu

Me ka mālama nui, a ma lalo o ka hooponopono ana o ka lapaau ia kekahi i ka hana o ka "Ksarelto" kauoha no ka hoʻohana (like analogues) i loko o ka kēia hihia.

  • malamaia lakou nei, e hoomanawanui i ka poe i ka māhuahua pilikia o ke kahe ana ke koko i loko o ke kahua;
  • nei Neʻe ulcerative maʻi me ka predisposition e relapse;
  • lapaʻau o kaʻaʻa puʻuwai 'ole e loli iki degere ma ka hui pu ana, me ka ai' i māhuahua rivaroxaban ka maʻiʻo ma ke kino o ke ahonui;
  • Hoʻomanawanui iki mai undergoing Inc ai 'hiki ke' ō hemostasis;
  • hoomakaukau i mea hiki ke hoʻoulu i ka nui o ka rivaroxaban, e laʻa me, antifungal ai 'AZ pūʻulu;
  • i ka lāʻau a me ka mea like papa "Ksarelto" ua contraindicated i loko o nā mea maʻi me HIV, ina pono ka mea, i kekahiʻano o ka protease nā mea kūpale o ka mea hoʻomaʻi.

Inu i hāpai keiki, a breastfeeding

I ka lā, ka mea, ua i kaʻoi loa paa, e like me ke keiki "Ksarelto" analogues o ka lāʻau ma ka hopenaʻoi loa a me ka maluhia ma ka hapai wahine.

Ho okolohua i mālama 'ia ma ka keʻena hoʻokolohua holoholona i hōʻike haʻi kaʻawahia o kaʻeleu waiwai o ka hoʻomākaukau i meaola expectant makuwahine, e like me ka lāʻau a nā loa reproductive kaʻawahia o ka wahine kino.

E like me ke keʻena hoʻokolohua haʻina, ka lāʻau "Ksarelto" mea like i ka mea like me ia i pharmacological 'ana i ka hiki e kela kapa o ke keiki, no laila, i ka lāʻau ua contraindicated.

Nō hoʻi i ka wā o ke noi ana o "Ksarelto" wahine e ole poina e pili ana i ka mana ana o ka contraception, mai ka hapai ana, a accompanies i ka wehe ana o ka lāʻau, hiki negatively pili fetal ulu.

Pahuhopu hoopai e pili ana i ke kanawai o ka lāʻau 'ia i loko o ka lactation au, i ka manawa hakuʻole, akā, keʻena hoʻokolohua haʻawina ma ka keʻena hoʻokolohua holoholona paipai i kaʻeleu waiwai - rivaroxaban - mai ka hiki e metabolize aʻaʻole excreted ma ka umauma o ka waiu. Nolaila, breastfeeding e haʻalele i ka hoʻohana 'ana i ka lāʻau.

Ma muli o kaʻikepili hoakakaia ma ke keʻena hoʻokolohua haʻawina, ua hiki ke olelo ia rivaroxaban aʻole e pili mai i ka hiki ana o ka kiʻie oʻo meaola e ho okumu viable keiki ma kaʻiole, akā, i loko o kānaka i kēiaʻano o ka ho okolohua i ua hana.

Pūnao a me ka hoʻopau alahele

No ka enteral? Eaia, he ekolu aoao o ke? Aneii, a hoʻopili like i kekahi hapakolu o ka huina helu o ka ole-metabolized lāʻau:

  • urinary excretion;
  • excretion i loko o ka feces;
  • hoʻopau Viaʻaʻa puʻuwai excretion laina (i loko o keia hihia, kokoke i waiwai metabolized a eliminated ma unmodified ano).

Biotransformation rivaroksaba hana ma maomeka i mea kuokoa o ka cytochrome nenoaiu.

Na ka papa kuhikuhiE alanui - ka'okesaside o ka morpholino pūʻulu a me ke anoe o ka amide paa ana me ka wai.

Haʻawina mālama 'ia ma ka lūmaua, ke manao aku nei au rivaroxaban mea i ke kumu no ka P-glycoprotein a me ka kumuʻiʻo e hoʻolako ia'ku oncological umauma maʻi.

Nō kāu, ana o metabolites ua lawe mai ma 5-9 hola.

ʻaoʻao waiwai

Ana e olelo mai ai i ka hoomakaukau kuhikuhi no ka hoʻohana: e e lawe analogues "Ksarelto" a me ka hoʻoponopono 'ka lapaʻauʻia wale nō ma luna kuhikuhi. Ke aʻo iho wehewehe i au mamuli o ka laʻau heluna o ka lāʻau, a me kona analogues. Mai poina i ka heluhelu i ke aʻo? Eaia!

Aia ma lalo Hōʻike 'ia nā mea a pau hua'ōlelo i keʻano o ka hanaʻana a me nā reactions a he lāʻau' "Ksarelto" analogs. Price huaale - mai 900 rubles. He inexpensive ka wā e noonoo i ka hapanui o kaʻaoʻao 'ole nā hewa i ka rula.

  • ʻaoʻao 'ole i i ua ike ka wā hoao ke koko a me ka lymphatic nenoaia, i anaemia, a thrombocythemia, a hōʻike infrequently.
  • Tachycardia - ka mea wale adverse naoh ka wā e lawe i kēia k.
  • Hemorrhage.

Eia na kumu i contraindications i ka lāʻau "Ksarelto" ke aʻoʻia.

Analogs o keia k hiki i ka malfunction o ka digestive'āpana: kahe ana ke koko, IIeEeAIEUIeXAIIUE eha, dyspeptic symptoms, i kekahi manawa - maloo waha.

Aie i ka hoike o rivaroxaban kūloko reactions ke kānāwai: wela, haanou ana ma ka ka pahu kui paena ka wā lawelawe parenterally iaoia, nawaliwali a me ka malaise.

Ka muli o kēia mau keʻano o ka hanaʻana he hoʻonui i ka hoomakaukau "Ksarelto" counterparts. Ke kumukuai o ka lāʻau ', like me ka rula, mea maʻamau ma nā mea a pau hale kūʻai lāʻau lapaʻau mau kaula.

Nā Papahana O Ka ho ohana a me laʻau heluna

Piha 'ana i ka pololei? Eaia hiki i ai i ka lāʻau kekahi loa "Ksarelto" ke aʻoʻia. Analogues o ka lāʻau i loko o kēia mau mea,ʻaʻole mea fundamentally okoa.

Kēia lāʻau i loaʻa ma ka papa palapala, no laila, Akala a ua lawe enterally. Inā ka hoʻomanawanui no kekahi kumu hiki ole ke ale wale iho i ka papa - ka mea hiki ke wāwahi ihola, a hui me ka kupono o ke kinowai (kī, ka wai).

Ma hope o ka loaʻa 'ia k ‰ e koke hahai i ka palaoa.

overdose

Ole e hooko me kūmau? Eaia "Ksarelto" hiki overdose, i ku una oia symptomatically, e like me ka lāʻau i ka maopopo antidote.

I mea e emi adsorption o ka lāʻau i loko o ka uuku liʻiliʻi hiki e kekahi sorbent, e like me ho'ā 'kalapona. No hoi e hōʻeleu i excretion o metabolites e pono ai, e hōʻike i ka lalau wale, diuresis, a ua lawe mai Via hoʻohana o ka nui dala o ka loli a me ka pono o diuretics.

kumukūʻai

Ke kaumaha ma muli o ka Hookah, ke kumukuai o "Ksarelto" lāʻau loli aʻe mai 899,00 rubles. no ka 10 na papa, i pihaʻi me 10 mg oʻeleu 'Oponopono, i 1740,49 hamo i.

Makua, i ka i 30 pellets, hiki ke kuai no 3300,00 rubles.

Ka nui loa AEeAaOA he 100 capsules, ka mea, na koina 8600 rubles.

Kumu kūʻai Policy "Pradaksa" lāʻau hilinaʻi nui ma luna o ka laupaʻi ka maʻiʻo o kaʻeleu 'Oponopono no mea hōʻikeʻikeʻuʻuku:

  • 75 mg - 716,00 hamo i;.
  • 110 mg - 1574,00 hamo i;.
  • 150 mg - 1676,00 hamo i.

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