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Benzathine benzylpenicillin: ano, ka waiwai a me ka noi, analogs

Benzathine Benzylpenicillin mea he antibiotic a me ka pili ana i ka penicillin pae. Hoʻohana 'ia no ka hana a pau ano o infectious mai, kena ae la ia e koʻohune susceptible i kona hana. Ma keia 'atikala, e hoonoho aku makou i mai i ka au mamuli o ka aʻo no ka pono, nāʻikepili a me contraindications i ka lāʻau', like me papa he mau na¯.

Benzathine benzylpenicillin: hōʻike ana i ka lāʻau '

Kēia lāʻau 'o kekahi o ka pae mua o ka penicillin antibiotics. I loko nō o ka lōʻihi loa kau noi, ka mea i ole nalowale kona pilina aie i ka laulā huahelu o ka hana, a me ka hiki, e pepehi i kekahiʻano o pathogenic koʻohune. Ka lāʻau, no kekahi laʻana, hiki Makuakane me anthrax, meningococci, syphilis a me ka ai iiiaanoaa o streptococci a me ka staphylococci. Ua injected like i loko o ka digestive'āpana ua i ke kemu benzathine benzylpenicillin.

Beauty ma Roma ua pinepine i hoakaka ia ma ka kauka, a laila, i ka hoʻomanawanui mea ole e maopopo mea kana i haawi mai ai. E pale i kēia ka hilahila, oe wale pono e ike i ka inoa o ka lāʻau i loko o kēia 'ōlelo - Benzathine benzylpenicillinum.

Nō kāu, i ka lāʻau 'ua lawelawe intravenously paha intramuscularly. Akā, he mea hiki a me ka lāʻau haawi i loko o ke kino ma ka spinal Canal, subcutaneously 'ole ma o ka loli ana o wahi.

Benzylpenicillin - antibiotic haku, mai ka ia hana waiwai. Akā, e komo i ka lāʻau i loko o ka palapala o ka paʻakai. Nolaila, o ka waiwai a ke waiho waho no ka lōʻihi manawa ole e wawahi ana ilalo. A ma hope o ka hoʻokomo 'ia' ana o penicillin G ua hookuu mai i ke kino o ka paʻakai, a hoʻomaka kona antibacterial hana.

Ke kaumaha ma muli o ka mea ma i ka paakai o kaʻeleu waiwai, i kekahi mauʻano o ka lapaʻauʻia. I loko nō o kēia, ka mea a pau i'ōlelo koʻikoʻi akulaʻo ia ia, a me kekahi mau 'ole o ka hooponopono a me ka lōʻihi o ke kanawai.

hoike

Benzathine benzylpenicillin ua hoakaka no ka mea i kēia maʻi.

  • Nā mea palahēhē o ka ÷ naehana hanu nā loko (pleurisy, pneumonia, bronchitis, empyema , a pela aku.).
  • Maʻi o ka genitourinary'ōnaehana (syphilis, gonorrhea, urethritis, cystitis, adnexitis, salpingitis).
  • Nā mea palahēhē o luna naehana'āpana (ula wela, tonsillitis, sinusitis, otitis Media, sinusitis, laryngitis, etc.).
  • Purulent nā mea palahēhē o ka pilikia makapō nā loko, na iwi a me ka ili, mucous membranes (ophthalmia, dacryocystitis, blepharitis, osteomyelitis, mediastinitis, erysipelas, cellulitis, wahi iho la maʻiʻaʻai, a pela aku.).
  • Brain abscess.
  • Purulent meningitis.
  • Septicemia, sepsis.
  • Arthritis.
  • Peritonitis.
  • Mai, kena ae la ia e spirochetes (yaws, anthrax, etc.).
  • Wela, kena ae la ma ka iole nahu.
  • Nā mea palahēhē kena ae la ia e Listeria, Clostridium, Pasteurella.

Eia kekahi, i ka lāʻau 'ua lawelawe i loko o prophylactically postoperative complications a me complications me streptococcal maʻiʻaʻai (endocarditis, rheumatic kuni, glomerulonephritis, a no laila, ma luna o.).

Pharmacokinetics

Benzathine benzylpenicillin (Lakina Benzathine benzylpenicillinum) koke ma hope o aaieieno? Hoʻomaka e disintegrate, ka hoʻokuʻu 'i kaʻeleu waiwai. I ka Ia manawa ka lāʻau i koe i loko o ke koko o ka ae 3 pule ma hope o ka ka pahu kui. Ke kinowai waiwai komo iloko o ka maikaʻi ma mua o loko o ka'aʻaʻa. It E e kaʻikaʻiʻia ma ka manaʻo i benzyl penicillin mea hiki ke lanakila i ka placental ke'ākeʻakeʻa mai, aʻikeʻia i loko o ka waiū o ka poe makuwahine. Excreted ma nā puʻupaʻa i loko o ua hoʻololiʻia palapala. Iloko o ka mea mua 8 lā hoʻokuʻuʻia ma kahi o 33% o ka lawelawe mahele lāʻau.

Hāpai keiki a me ka umauma-e ai ana

I kaulana ma luna, i ka lāʻau mea hiki ke komo iloko o ke keiki, a komo i loko o ka umauma o ka waiu. No laila, e ke hele breastfeeding ka wā ka lawelawe ana i ka waiʻona.

Ma hāpai keiki, ke kohoia ana o ka lāʻau mea hiki wale ina o ka pono no ka wahine, ua oi aku ia mamua o ka ka pilikia no ke keiki. Ke hoʻoholo Pono e i e kekahi kahuna lapaau, ao wā e hiki mai makuwahine e pili ana i nā mea a pau i ka hiki hopena.

Contraindications

Benzathine benzylpenicillin (beauty e koi 'ia kekahi kauka) i ka helu o contraindications. Ka mea, e ole e hoakaka ia ke kanaka me ke kēia illnesses:

  • Intolerance e penicillin paha cephalosporin, he allergic naoh ia ia.
  • Ke kiʻekiʻe nui o potasiuma i loko o ke koko (hyperkalaemia).
  • Arrhythmia.
  • Hay kuni.
  • Bronchial asthma.
  • ʻaʻa puʻuwai insufficiency.
  • Pseudomembranous colitis.

Kaiapuni medicament lawelawe i na keiki i ka eono mahina, a prematurely.

ʻaoʻao waiwai

Benzathine benzylpenicillin hiki i kekahi undesirable loa, helu ia ma lalo iho nei.

Ke Kula Kaiapuni 'allergic reactions:

  • kuni;
  • hives;
  • wawe ma ka mucous membranes a me kaʻili;
  • ami eha;
  • eosinophilia;
  • erythema multiforme;
  • Angioedema;
  • exfoliative dermatitis;
  • anaphylactic kŰia.

Adverse reactions o ka mea'ōnaehana mānowai koko'ōnaehana:

  • thrombocytopenia;
  • anemia;
  • coagulation kāna hana;
  • leukopenia.

Eia hou:

  • stomatitis;
  • headaches;
  • glossitis;
  • ʻeha i loko o ka wahi o ka hooponopono;
  • abscesses;
  • infiltrates;
  • jadeʻike ākea;
  • fistulas.

Me ka hooloihi ae i hoʻohana ana i nā palapala fungi a me anakahi iki-meaola ke ulu ia'ku, laila, i ka lāʻau, e lilo kona laulā.

Benzathine benzylpenicillin: kauoha no ka hoʻohana

E hoomanawanui i mua o 12 makahiki, i ka lāʻau 'like me ka kāohi ana a me ka hana ana o infectious maʻi ua lawelawe hookahi o ka hebedoma i ka laʻau heluna o 300 a hiki i 600 tausani. Units a palua ka mahina ma 1,2 miliona huahelu.

Like kāohi ana no ka rumatika mea oioi laau no 6 pule, hookahi manawa i ka pule a hiki i 600 tausani huahelu. I ka Ia manawa i hoakaka ia aspirin 'ole' ē aʻe NSAIDs.

Hoʻomanawanui iki mai kaikaina ma mua o 12 makahiki, i ka lāʻau 'ua lawelawe hookahi o ka hebedoma i ka uku o ka 5-10 tausani. Units no 1 kg.

Ma waena o injections e lawe wahi ma ka liʻiliʻi 8 lā. Ka awelika laʻau heluna o 2.3 miliona 'iniha, kapuaʻi.

Mua ana, i mea hoʻoheheʻe ka lāʻau i loko o Saline, ka wai no ka pahu kui a hoc ole novocaine (2.5% a 5%).

Hoʻolauna i ka lāʻau e ia i loko o ka kēiaʻaoʻao:

  • intramuscular;
  • intravenous;
  • subcutaneous;
  • Lumbar (Via ka spinal Canal);
  • pleural (ma ka pulmonary pleura);
  • subconjunctival (Via ka ocular nā'aʻaʻa);
  • drip ma ka pepeiao;
  • drip ma ka ihu;
  • 'ana i ka loli ana o hui,'aʻaʻa.

Ka hui pu ana me ka 'ē aʻe ai'

Benzathine benzylpenicillin (aʻo 'ana e like me ka hōʻike) e pāʻani aku me nā ai'. Pela oia i benzylpenicillin e i ka i kēia mauʻanuʻu: he synergistic, antagonistic a me ka bacteriostatic.

Eia hou, i ka lāʻau maoli ka laulā o ka ai ', no i kaʻauhau'ēʻaʻe anticoagulants. A ho'ēmi i kā ka laulā o ka ethinyl estradiol a me nā moʻolelo contraceptives.

E hoʻohana pū me NSAIDs, allopurinol, diuretics i nā hualoaʻa ma ka ho'ēmi i kā omo secretion, a māhuahua nā hoʻohui like oʻeleu 'Oponopono. Eia hou kekahi, allopurinol nui maoli ka pilikia o allergic reactions.

precautionary ana

Pono ma mua o ka ka pahu kui mua ka pono i ka aspirate. Inā ka lāʻau accidentally loaʻa i loko o ka ipu koko, ka mea hiki i ischemia paha embolism. Eia hou, aia i e ka manao o ka iini, kaumaha, transient blurred hihio.

Ma na wahi e pono e hana mau injections i kekahi manawa, i ka lāʻau 'ua lawelawe ia ma kekahi lima a me kīkala.

Ka wā pono e keʻakeʻa koke na hoikeana mua o allergic Inc. E like me ka noho ana i ke kauka i hoakaka ia Allergy lāʻau.

Pinepine me ka benzylpenicillin hoonoho i "Levorinum" a me "Nystatin", me he mea i ka pilikia o fungal nā mea palahēhē. He nolaila lōʻihi-manawa Inc ka lāʻau kānāwai inhibition o intestinal microflora i paha ke nā wikamina B. Ma keia manao, hiki ke lawelawe i ka intramuscular hooponopono o kēia nā wikamina.

Cautions

Benzathine benzylpenicillin ia me ka mālama nui i loko o nā mea maʻi i i malama i keʻano o ka hakuʻala hana, he mea he predisposition i allergic hoike ana, me ka kiʻekiʻe pā lonoaʻili i ka hana 'Oponopono. I ka manaʻo hoʻoholo i mauʻanuʻu me ke kahuna lapaau, ka mea e ike i ka mōʻaukala o Isaaka.

'Aʻole i paipai lāʻau no ka iapaau ana o neurosyphilis, mai keia maʻi hiki ole ke loaʻa ka makemake lehulehu o kaʻeleu waiwai ma ka hoʻomanawanui ka koko.

analogs

Aia nō 'ē ai' e i ka ia kanawai me benzathine benzylpenicillin. Analogs, o ka papa, i hui ole ia me ka penicillin pae. E helu i ka loa kaulana pono, a:

  • "Gramoks-D" - ua hua mai i loko o ka palapala o ka lepo i manaoia no ka? Aneii a me ka moʻolelo hooponopono.
  • "Amosin" - ua hua mai i loko o capsules, papa a me ka lepo no ka moʻolelo hooponopono.
  • "Maʻi puʻupuʻu" - ua i loko o ka palapala o ka malakeke.
  • "Hikontsil" - i loaʻa i loko o ka palapala o ka lepo a me ka capsules no ku una hooponopono.
  • Azlocillin paʻakai paʻakai - me ka pauka, waiwai, mai a e ka pāʻoihana no intravenous ka pahu kui.
  • "Ampicillin" - Ua loaʻa i loko o na papa, capsules, granules, ka polokalamu e ka slurry, a ua laweʻia hōʻike waha.
  • "Ekobol" - hua papa.
  • "Ospamoks" - ua i loko o ka palapala o ka papa, capsules a me ka lepo no ka moʻolelo hooponopono.
  • "Phenoxymethylpenicillin" - Ua loaʻa i loko o na papa, dragees, granules, a me ka pauka.
  • "Star-Pen" - ua i loko o ka palapala o ka granules, a i nāu kekahi, a lawe hōʻike waha.
  • "Oxacillin" - ua i loko o ka palapala o ka papa, capsules, he lepo lā, mai a, i ka pāʻoihana no ka pahu kui.
  • "Standatsillin" - Ua loaʻa i loko o capsules.
  • Carbenicillin disodium paʻakai - ua hua mai la i ka pauka ano no ka hana ana o ka pahu kui pāʻoihana.

Penei, hoʻowahāwahā ka kŘpa a lōʻihi-makahiki i o ka lāʻau ma ka lapaau, oia no koe kekahi o ka loa ka hoʻokō konohiki e ku ei keʻano o nā mea palahēhē.

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