Ola kinoHoomakaukau

"Esomeprazole": aʻo no ka hoʻohana 'ana, maoli counterparts

"Esomeprazole" - he lāʻau e pili ana i ka Organotropona gastrointestinal ai '. Ka lāʻau i antiulcer hana a me ka mea i proton EII ni inhibitor.

I ka haku mele 'ana, i ke kalaʻana aku palapala "esomeprazole" lāʻau

Ka lāʻau 'Ua loaʻa i loko o ka palapala o ka papa me ka laʻau heluna o 20 a me 40 mg oʻeleu' Oponopono esomeprazole, e like me ka ano o ka lepo i manaoia no ka pāʻoihana no ka pahu kui (40 mg hue). Lole komoʻuʻuku nona na papa, noho male 'ana a lawe wahi i loko o ka naʻau liʻiliʻi.

Pharmacological hana "esomeprazole" lāʻau

He aha mea i ka lāʻau "esomeprazole"? Na Ke Kumu no ka hoʻohana hōʻike i kēia antiulcer konohiki, a, i ka nawaliwali kumu, oia ke launa i kaʻeleu palapala ma hope, inu. "Esomeprazole" inhibits ka'ūhū H + -K + -ATPase haʻawina, a me ka secretion o hydrochloricʻakika (hauma¯na, basal). Pono 'ana ia lŘlŘ loko o ka hola ma hope o' ai, inu o ka lāʻau. I ka loaa ana "esomeprazole" i kela la i keia, no ka lāʻelima, i ka allowable kela la i keia mahele lāʻau - 20 mg ma hope o stimulation ma ka pentagastrin i kā mākou kiʻekiʻe o hydrochloricʻakika ua hoemi kūpono kou (ma kahi o 90%).

Pharmacokinetics

"Esomeprazole" kauoha no ka hoʻohana mea like me ka lāʻau i, penetrating i loko o ke kino, hoʻomaka koke a me ka pono o ke kemu, e hoopaa ana i nā polokinaʻaneʻane 100% (97%). Ke bioavailability māhuahua me ka hana hou 'ia' ana o ka lāʻau, mai 64 a hiki i 89%. Ke medicament i ka palapala ana o metabolites a excreted kuhikuhi ma ka mimi, He nīnūnē hapa o ia mea noho i loko o nā feces.

Nāʻikepili "esomeprazole" hoomalolo

"Esomeprazole" analogues hoʻohana i nā mea maʻi me ka gastroesophageal reflux maʻi lapaau a me relapse Kāohiʻana. Ke hoʻopololeiʻia ana ma ka iapaau ana o ulcers o ka opu a me duodenum, no ka pale maʻi i kupu mai ma muli o ka NSAIDs.

Ke k hoʻohana ma peptic ulcer ka wā loli duodenum a me ka'ōpū. Ua hiki ke hoopili i ka hoʻomanawanui iki mai ka poe i ua hoola esophagitis, iloko o hooloihi ae i relapse Kāohiʻana. Ana ami palapala noi me nāʻano "esomeprazole" antibacterial ai '. Papa a me ka pahu kui i loko o ka luna 'Inc ma keia hihia ae luku Helicobacter pylori.

Contraindications i ka loaa ana "esomeprazole" lāʻau

Contraindications nā makahiki emi o umikumamalua makahiki, hypersensitivity e esomeprazole, i ka wā o ka breastfeeding. Ka hopena o ka lāʻau lapaʻau i ole, ua hoʻokumu 'ia i hāpai keiki.

lāʻau'Āpana

Ka lāʻau 'Ua hoʻohana i ka kela la i keia mahele lāʻau o 20-40 mg. Ka lōʻihi like 'ole o ka Inc me ka nānā' nāʻikepili regimen a? Eaia ka hoʻokōʻana medicament "esomeprazole". Papa a me ka paakiki waikahe e kākoʻo pāʻoihana maʻaʻa puʻuwai insufficiency ka hoʻohana 'ana i kā mākou mahele lāʻau o 20 mg.

Erosive reflux esophagitis kamailio ana no eha pule me ka kela la i keia mahele lāʻau o 40 mg. Ma hooloihi ae i Kāohiʻana o ka recurrence ma muli o ka loaa ana o ia hoʻi, he hoomanawanui ma i esophagitis i ua ola, i ka i kela la mahele lāʻau ua hoonohoia ma ka laulā o ka 20 mg.

Ma ka iapaau ana o ka reflux oesophagitis, nona ma kamaʻilio akula i ka hp'pnphp maʻi symptoms, lawe 20 mg o ka lāʻau "esomeprazole". Hoomakaukau i loko o ka palapala o ka papa, a he lepo lā ua hoʻohana 'ia e pepehi H. Pylori, ka wā he mea kamaʻilio me duodenal ulcer, i loko o ka hoʻohui pū Inc - "esomeprazole" (20 mg), "Clarithromycin (500 mg)," amoxicillin "(1 g). A pau ka lapaʻauʻia ia i nā manawaʻelua i ka lā.

'ōpū ulcers kena ae la ia e NSAIDs, ka mea, ua? Aeiiaiaoaony e hana 20 mg "esomeprazole" no ka lā. Ke makemake mahele lāʻau ua mau ia i ke kahuna lapaau e pono e lawe i ka mooolelo o ka ola o ka hoomanawanui, i ka maʻi, me ka oolea o kona papa, a me kekahi mau aʻe.

ʻaoʻao 'ole "esomeprazole" lāʻau

E hoomanawanui i ka poe i lawe i kēia mau ai 'no ka lōʻihi manawa, ua oi prone i ke kahua o ka glandular cysts i loko o ka'ōpū ma mua o nā nā mea maʻi. Ka loa pinepine adverse hoike ana o ke kino i iapaau ana o ia hoʻi, "esomeprazole" aʻo ma o ka palapala noi allocates he headache a me kekahi hopena maikaʻi reactions mai ka gastrointestinal'āpana, e like me: constipation, flatulence, diarrhea, nausea, ka luaʻi, imua o kaʻeha i loko o ka abdomen. Ma rarerʻaoʻao 'ole nā ka maloʻoʻana o ka mucosa o ka waha, pōniuniu, urticaria, ka ohane, dermatitis. e hiki Other reactions, no laila, pono e lawe i ka iapaau ana mai ikaika ma lalo o ka hooponopono ana o ka hoʻomalu.

Overdose ua pu e mau nawaliwali, e māhuahua mea hiki wale mai o kaʻaoʻao waiwai, a me ma ka aoao o ka digestive'āpana. Ma na hoopii, lapaʻau ua hana ma ke kāpaeʻana i nā symptoms o overdose a me ka mālama 'ana i Inc. Dialysis i aneane i makemake ai, aole he antidote.

Cautions

Hapai wāhine "esomeprazole" analogs lawelawe me ka lōʻihi mālama nui. Lapaʻau i hāpai keiki e e kākoʻoʻia e ke kauka. ka lāʻau 'ua kuhikuhi i hapai wahine wale ma ia mau hihia a pau ma ka maikaʻi hopena o ko lākou mau kino me ka nui loa aku i ka Loaʻaʻiaʻino i ka unborn keiki. Ike loea ikepili ma ka hopena o ka lāʻau ma luna o ka embryo mea i keia manawa, a hiki i hiki e pale aku lapaʻau me keia ka lapaʻauʻia. E ho ohana ana o ka lāʻau "esomeprazole" ka wā umauma-e ai ana ua pāpā.

I ka mea 'aʻe' ana i ke akepaʻa loa i ka ahaaina i mahele lāʻau hoʻopōʻino i ke ola (ina mau aʻe 'ana e hoʻoponopono).

I ka wā o ka hoʻomanawanui i ka symptoms i wae neaiae, e like me hematemesis, dysphagia, nausea, nui ka ho'ēmiʻana i loko o ke kino paona i ka iapaau ana au "esomeprazole" i mea e hoʻopau ai ulcer no i lawe i ka lāʻau i loko o ke alo o ke kēia maʻi, malignancy E e holoiʻia. E kuhikuhi i ka malignant ano o ka hikoko mea pono e hoʻomaka i ka mahele.

E hoomanawanui i ka poe i ka nele o ka sucrase-isomaltase, hereditary fructose intolerance pūʻulu papaia e koho "esomeprazole" synonyms.

AaOIeIOUIeXAOAaIN "esomeprazole" me nā ai '

Me ka mea i ka wā hoʻokahi pono o ka lāʻau a me "citalopram", "clomipramine", "imipramine" e hiki potentiation o kēia mau Luna,? Ienoai o kaʻeleu waiwai i loko o ke koko. Wā hoʻohana i ka huipūʻana me "esomeprazole" hoemi ka hoʻokōʻana "ketoconazole" "Itraconazole" worsens lākou omo.

I ka hoʻohuiʻia o ka "esomeprazole" me "ATV" Ua Ua he nui emi i loko o ka waiū o keia k. "Esomeprazole" pae'ōnaehana aʻoʻia,ʻaʻole pono e hoʻohana ka poʻe me ka "phenytoin", "clomipramine", "imipramine" a me ka ai 'e like me "citalopram", "Diazepam", "Nelfinavir" a me ka "Atazanavir". Ka nui o kēia mau ai 'mea hiki ke ala i loko o ke koko, no laila ia i ohiia, e emi lākou nā māhele. Concomitant ana o «esomeprazole" a 'o ia hoʻi "clarithromycin" hiki aku i ka lula' loli ma ka waiū "esomeprazole" mākaukau kaua paha ma mahuahua kona pili me ka inhibition o pūnao o ka lāʻau. A E e akahele manaoia instrukiyu i ka lāʻau a me ka nīnau aku i ka hoʻomalu.

Ke kumu o ka lāʻau, hōʻike manaʻo e pili ana i ka lāʻau "esomeprazole"

Ka lāʻauʻano nui loaa ma ka papa palapala. Keʻena kūʻai lāʻau lapaʻau "esomeprazole" hiki ke loaʻa ma lalo o ka oihana inoa "Nexium" a me ka "Emanera". I ka wa e kuai i ka lāʻau "esomeprazole" kumukuai hilinaʻi nui ma luna o ka mahele lāʻau o ka mea hana waiwai i loko o kona haku mele 'ana. Ke kumu o ka lāʻau ma ka laʻau heluna o 20 mg ( "Emanera") mea e pili ana 500 rubles. no ka 28 o na papa io, a me ka nānā 'ana i ka Hookah. Ka lapaʻauʻia me ka mahele lāʻau o ka 40 mg o ka hana 'Oponopono ( "Nexium" 28 papa) hiki ke kuai no 3000 rubles.

"Esomeprazole" i hōʻike manaʻo ka hapanui maikaʻi. Ka mea, uaʻike ka lāʻau waiwai e inhibitʻakika secretion, nā basal a hauma¯na. Ka lāʻau 'Ua hōʻike kiʻekiʻe hopenaʻoi loa i loko o ka iapaau ana o ka olelo e like me nāʻikepili i hoakaka ia ma ke aʻo. Ma Inc, ia 'o ia hoʻi he mea he hōʻemi iki pahiki o kaʻaoʻao loa. 'Aʻole i pau ka hiki wawe ka hiki ke loaʻa i ka lāʻau i loko o keʻena kūʻai lāʻau lapaʻau, kekahi e hoomanawanui i ka poe i loaa "esomeprazole", ke kumukuai manao kiʻekiʻe.

A o ka poe i ka lapaʻauʻia i hoakaka ia ma kekahi kauka ma hope o ka kūlike loa ka wehewehena o kaʻike, a me ka paipai mahele lāʻau, e koho i ka nui hana i loko o ola. E like me ka nāʻana, "Nexium" ka poe hanohano i waena o nā mea maʻi ma mua o "Emanera". I ka "Nexium" gastric hoʻolako i ke ano o ka makemake hopena ma hope ma kahi o kekahi mahina ma hope o he lālā o ka Inc. Ka hoʻomaikaʻi i ke ano hiki ke'ākoʻakoʻa ma hope o 1.5 pule o ka nohoʻana. ʻaoʻao 'ole i loa pohihihi keia. Uluwehi O "Nexium" ka hoʻokō, ka mea e kokua me ka hoʻopau o nā kūlana haawiia i loko o na kuhikuhi. I ka hopena ua 'oluʻolu, e mea pono e hoʻokō' ia i ka papa holoʻokoʻa, a hoopau hoopili aku i ke kauka i ka koi.

Analogs "esomeprazole"

ʻO kēia mau koho hiki ke ike okoa mai analogues o ka lāʻau.

  • "Omeprazole" - i kapaia "Losek", "Omez", "Ultop";
  • "Rabeprazole" - he makaukau iʻikeʻia ma lalo o ka inoa "Ontaym", "Zulbeks", "Noflyuks" "Pariet", "Hayrabezol";
  • "Pantoprazole" ( "Sanpraz", "Kontrolok", "Nolpaza");
  • "Lansoprazole" ( "Lanza", "Lanzoptol").

mau ai 'a pau i like' ole, akā, e oko mai kekahi i kekahi i loko o kā lākou waiwai.

Kulike "esomeprazole" a me ka "Omeprazole". Oko o kēia mau ai 'i maopopo. "Esomeprazole" mea he isomer "omeprazole". Kēia la hoomalolo, e hoʻomaka ana mai o ka 'inikua moʻokalaleoʻikepili, ua he nui ia Morohiha, akā, he like hana o medicaments. "Omeprazole" mea he lāʻau kumukahua waiwai i ka helu nui o kaʻaoʻao loa. Inā i ka waiwai o ka "esomeprazole" mākou noonoo, i ka lāʻau 'ua hooku iho la ia me ka hoonui ae i hoʻokolohua o "omeprazole", ke kumukuai o ka a i o Laielohelohe he nui nā mea maʻi. Eia naʻe, "esomeprazole" emi paha e i hua'ōlelo i makemake reactions, no laila kona kūʻai ua noʻonoʻo oi waiwai ma mua o kūʻai "Omeprazole".

"Rabeprazole" a me ka "esomeprazole" i ka like Nine Inch haku mele 'ana, ka mea hana i ka ia maʻi. Akā, poe akamai i manaʻo i loohia i kekahi, e like me gastroesophageal reflux maʻi, "Rabeprazole" eliminates oi ka pono, ka mea e lawe aku oe i ka symptoms maikaʻi, e ka poʻea pau i ka kokololio loaa o ka esophagus hana. I ka nele o ka maikaʻi hookoia ma ka iapaau ana o "esomeprazole" i e pili ana me na ano kanaka o ka meaola.

Inā pono, koho i ka mea like, e nīnau aku i ke kauka. Hana hou lehulehu i ko lakou ola, a me kekahi, e nana i ka manawa, a laila, ke loaa e e wikiwiki a me oe, e pale aku i na complications.

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