Ola kinoHoomakaukau

Alpha-blockers: hōʻikeʻano a me ka Mea Maluna

Mahalo i ka 'epekema noiʻi i loko o ke kula o pharmaceuticals ua mau aʻo i ka hana o ka ai', ke kala o ka oi kēia kiʻekiʻe-hana ai '. Akā, he mea ai 'he ākea huahelu o ka hana i ka mea paʻa mau no ka makahiki. Mau nā Alpha-blockers.

Loa pinepine ka mea, e hoʻohana 'ia ma ka lāʻau lapaʻau o hypertension, no ka hakumakuma ke koko, e like me ka helu o urological kāna hana, e laʻa me, maʻi prostatitis a me benign prostatic hikoko.

Mōʻaukala o ka Kaka

I ka loaʻa o ke Alpha-blockers ma ka Lūkini mea lāʻau lapaʻau hana ia i loko o ka makahiki 1976. No ka mea, ua noonoo lakou i ka hoʻokō ai 'a ho'ēmi i ke koko,. Akā, kā lākou hoʻohana mea,ʻaʻole manawa kūpono no ka mea, o ka nui loaʻaoʻao ole. Kekahi o na ai 'mua o keia pae ua "Prazosin". Next, ka mea i ee? Iecaianoaaiiuo o nā Alpha-blockers e like me "Doksasozin" a me ka "Terarozin". A pau o ia mau mea, e like me ka pono me "Prazosin", hoʻohana 'ia e pono hypertension, akā, i kekahi, mai ka mea oi hooloihi ae i hana.

Akā, i ka oko ao ma ke degere o ka IIeEeAIEUAA o ka wahi, a me ka ooieoeiiaeuiiai manao o Alpha-blockers. Hoomakaukau e e hōʻike mai iā ia ma lalo nei.

ano

Adrenergic receptors e māheleʻia i loko o nā subspecies:

  • Alpha-1 receptors, a i IIeEeAIEUIeXAIIUE ma luna o ka ili o kaʻili lahilahi o ka postsynaptic neuron, kuleana no na lepa lawe mai ma ka hoʻohana 'ana i ka helu wahi'ē aʻe catecholamine neurons a effector keena, a me kekahi mau vascular keena. Ke no o ka ha awina o kēia mau receptors mea vasoconstriction.
  • Alpha-2 receptors, a i aia ma luna o kaʻilikaiʻili lahilahi o ka presynaptic neuron ke kāpiliʻana hanauna o norepinephrine i loko o ka mauae synaptic i kekahi io manaʻo, ma laila hoemi i ka? Iecaianoaaiiie o noradrenaline, loaa i loko o ka mauae synaptic.

Manaʻo mea loaʻa blockade o Alpha-1 vascular ala apuupuu Muscle vasoconstriction eliminates hoʻonāukiuki catecholamines. I ka huli Alpha-2 receptors aia ma luna o ka presynapticʻili lahilahi o ka neuron,ʻaʻole blockaded, alaila, he mea pono no i ka manaʻoʻano papa hana, e hoʻonāukiuki i ke kala o ka noradrenaline.

E wae 1 (blockers) i hakaka o postsynaptic receptors. Oia medicaments hoʻopau mea loaʻa ha awina no a hiki i ka hopena o catecholamines kuu i ka holo, a me neurons.

oihana

Eia hou kekahi waiwai ma ke koko, ka ho'ēmiʻana, alpha blockers (ai 'helu' ia ma lalo nei) i'ē aʻe i hana '. Etokardialnye, metabolic, extracardiac pākōlea 'ole. Sci kiʻekiʻe ka hoʻokōʻana o keia pae ana o ai 'i loko o ka iapaau ana o ka loli ma ka myocardium, coronary nenoaiu, i ka mea e pono ai nā polokina i loko o ka prostate.

extracardiac

  • Stimulation o nā puʻupaʻa.
  • Hoomaemae ana o ka bronchial paipu.
  • Hou ana o metabolic keʻano o ka hanaʻana i loko o ka urogenital'ōnaehana ma prostate benignʻeho.

Alpha-blockers i he maikaʻi ia ma hoemiʻeho ka ulu a me ka degere o ka oolea o ke impotence.

cardiac

  • Ka ho'ēmiʻana o myocardial hypertrophy.
  • Hooponopono naau pāpana.

Me ka mālama nui no ka mea, o ka mea io ole, ua hoʻohana 'ia i loko o ka naʻau o ka hoʻokō' ole a me ka angina.

metabolic

  • Emi i ka pilikia o ka naʻokoko plaques.
  • Ho'ēmi i ke koko kō pae (insulina) i loko o ke koko.

E like me ka olelo ma luna, pinepine Alpha-blockers hoʻohana ma o ka iapaau ana o ka maʻi o ka prostate gland i loko o nā kānaka.

Ke kane kanaka ma luna o ka makahiki o ka 50 makahiki, pinepine ae aku, mai kēia 'ano o ka maʻi, i ka mua o ka a nō ka prostatitis a me ka prostate adenoma.

Kēia mau maʻi i ka hopena maikaʻi 'ole ma o ka kanaka o ka I Aloha Hawaii me ka a pau. Paakiki pilikia me ka urination, discomfort, e holumua ai impotence i kekahi mau hihia no na kanaka o kekahi makahiki. Eia hou, e noʻonoʻo ka luna-i oleloia mai e ke booming. Pinepine hiki ole ke hana meʻoki kino. E pau ana i ka maʻi huʻi pae i hoʻohana ai '.

No ka 'inikua' uao ua hoʻohana 'ia ka-blockers, nā mea kūpale o 5-Alpha-reductase.

Noaia pākōlea hana nā mea kūpale

I ka ulu ana o Muscle'aʻaʻa i loko o ka prostate ua triggered kuhikuhi hormonal. Steroid 5-Alpha reductase ka paipai 'ana i ka lua i loko o ka prostate gland hōmona testosterone hou' i loko o dihydrotestosterone. Ka hope, i ka huli, e hoopaa ana i ka nukelea androgen mea loaʻa i loko o ka prostate gland a stimulates ka secretion o paracrine ulu kumumea, ka mea, e hoi neʻe maila i loko o ka prostate. Alpha-blockers, e hiki ke kōkua i loko o kēia kahua nā mea kūpale o 5-Alpha-reductase.

Excessive? Iecaianoaaiiuo o dihydrotestosterone kumu i ka helu o ka loa e like me maʻi benign prostatic hypertrophy, Ka maʻi 'aʻai hikoko, prostate'ē aʻe urological maʻi. Ma kēia wahi i loko o ka hoʻohana 'ia nā mea kūpale o 5-Alpha reductase nā mea kūpale me ka' inikua lapaʻau papa. Lākou pākōlea hopena o ka blockade reductase, a ma ka huli emi na pae o DHT, i ke kumu no eiei? Prostate loli.

Ka loa Popular ai 'i loko o kēia hui e "Finasteride" a me ka "Dutasteride". Ka mea, i kekahi like pākōlea hookoia, oko waiū manawa a me ka regimen.

Blockers, hiki ke kuai nā mea kūpale o 5-Alpha-reductase ma ka hale kūʻai lāʻau lapaʻau ma kuhikuhi.

Akā, ma ka naʻe o ka ka hoʻokōʻana kiʻekiʻe, ai 'hoʻohana me ka mālama nui a me ka ole i na hihia a pau no i ka helu nui o io hoikeana a me contraindications.

Majorʻaoʻao waiwai ana ka lawe

  • Ma hope iho o ke ano o ka ai 'ana i lalo, ke koko, hoʻoneʻe' ia paha i ka hypotension.
  • Nausea, headaches a me ka pōniuniu.
  • Heart palpitations, pokole o ka hanu.
  • Muscle eha, nawaliwali.
  • Sedation.
  • Loli ka mālama, edema.
  • Pain i loko o ka'ōpū a me ka naʻau liʻiliʻi.
  • Ihu, pokole o ka hanu, makewai.
  • More pinepine ia i loko o ka wahine hapalua o ka heluna kanaka ua malama stimulation o bladder nawaliwali, pinepine urination.

No laila, e ke hoʻohana Alpha-Hoʻokolohua blockers me ka mālama nui.

Kekahi o na hopena loa hoʻoponopono mea postural hypotension, a e lawe wahi mua i hookahi mahele lāʻau. Kona symptoms hōʻike mua ma hope o ka hapalua o ka hora a me ka hola ma hope o ka loaa ana medicament. Ua piliʻano nui i "prazosin". E pale aku i kēiaʻaoʻao hookoia, ka lāʻau ai e haawiia mai ma ka ulu regimen a me kaʻoi loa i ka pō.

I e pili ana me ka luna i oleloiaʻaoʻao hopena o ka, alpha blockers koi 'ia ma ka hui pu ana me diuretics, e pale aku loliʻana a me painkillers e höʻike aku ka eha symptoms.

Medicaments o keia pae ua häʻawi mai me he kuokoa lapaʻau a me ka poʻe me ka 'ē aʻe lapaau no ka hana maikaʻi kela maʻi.

maʻi

Mau maʻi, no ka iapaau ana o ka i Alpha-blockers i hoʻohana:

  • Ma ka mana o ka hypertensive ka maʻi ma ka pu ana Inc like me ka mea e loaʻa ai kokololio pākōlea hopena.
  • Benign ka ulu o ke ana ma ka prostate gland.
  • Mimikō mellitus.
  • Pheochromocytoma.
  • Malignant neoplasm o ka prostate gland.

Contraindications

Ma ka hihia mai i hoakaka ia alpha- a me ka Hoʻokolohua-blockers?

I ka papa kuhikuhiE contraindications no ka loaa hoomakaukau ana i:

  • haʻahaʻa ke koko;
  • dehydration;
  • Inc me diuretics;
  • kela cardiac malformations;
  • maʻi naʻau ole;
  • asthma;
  • naau pāpana ka haunaele.

Mai Mai koi 'ia ai' o keia ano keia ano i gestation a me ka manawa lactation, e like me ka mea kūlike loa keʻena hoʻokolohua haʻawina ma luna o keia kumuhana i ua hana.

Alpha-blockers adenoma

Walaʻauʻana ai 'o keia pae e hoʻohana no ka iapaau ana o ka adenomas:

  • "Uroksataral".
  • "Cardura".
  • "Gitrin".
  • "Rapaflo."
  • "Flomaks".

Ma kekahi Alpha-blocker ka lapaʻauʻiaʻikepili. Ka papa hele ma.

ʻano papa hana o ka hana

Keʻano papa hana o ka hana ana i kēia mau ai 'i loko o ke kaua e kū'ē i adenoma mea puni, e lawe i ka leo o na nāʻiʻo o ka prostate a me ka bladder, pela kōkua e alleviate urination.

I koi 'ia ka lapaʻauʻia lapaʻau pololei me kanaka laʻau heluna, e lawe ana i kekahi paha mau manawa o ka lā.

I koi 'ia ka lapaʻauʻia nā waeʻano nā mea maʻi me ka holomua maʻi ka poe i pilikia me ka urination, a me ka nawaliwali ai' e ole i ka mea i makemake ia.

I ka papa kuhikuhiE pākōlea hookoia hoʻomaka e hele mai ma hope o ka pule o ka lapaʻauʻia. I 14-21 lā ka mea, he nui no ke kokua ana i ka hoʻomanawanui.

Cautions

No ka kiʻekiʻe pākōlea hopena i loaa i loko o ka paʻa o ka Alpha-blockers a me nā mea kūpale o 5-Alpha-reductase. Ke kiʻekiʻe ka hoʻokōʻana o ka i o ka hui kaulua hoʻomākaukau loaa like me ka hopena o ka 'inikua lapaʻau haʻawina.

Ua UaʻAʻole pono e hui pu iho i ka luna lapaʻauʻia concurrently me ka ai 'ole BADami impotence. E hiki anei i ka hōʻoi 'i ka pākōlea blockers kanawai, i mea undesirable. ʻO ka hopena o ke e kaʻoi emi i loko o ke koko,.

Kekahi hopena maikaʻi no o ka hooko ana o ka, alpha blockers Urologicals ejaculation e ia i loko o ka lua o ka bladder. Ua ke kumu ole io hopena no ka nohona ma ola.

I ka hoʻohana 'ana i kēia pae o medicaments no ka paioʻana adenoma paipai e emi' ē aʻe ai 'i ke koko,. Maliuia mai me he hehee ai o ka luna 'Inc, ka mea, i e emi kona mana ma ka iapaau ana o ka hypertension.

No nā mea maʻi e loaa ana mai ka hypertensive maʻi ana me ka loli ma ka prostate gland Alpha-blocker wā ua? Aeiiaiaoaony e noke kanaka hoʻoponopono i ke koko, pae.

Kaiapuni wā lawe ai '

  • Na laau me ka Alpha blockers e hoʻohana wale i hoakaka ia ma kekahi kauka. Ke kahuna lapaau e pono e ho oholo i ka mahele lāʻau, ka lōʻihi like 'ole o ka? Eaia.
  • Lapaʻau me kēia mau ai 'ia ma lalo o ka hooponopono ana o ka lapaau a' inikua Hoʻonaʻauao ma ka pā pōhaku.
  • A hiki i ka hoike ana o kaʻaoʻao 'ole e lawe i ka lāʻau, e ku malie, a nīnau aku i ke kauka.
  • I ole hihia e ole hoʻololi i ka laʻau heluna luna kū kaʻawale.
  • Other lapaʻauʻia ka poʻe me Alpha-blockers, e pili ana me ke kauka.
  • Mai hoʻohana Alpha-blockers me ka pōpilikia e Inc no hypertensive kāna hana me ka ae ole o ke kauka.
  • Maiʻae lā ai 'a hihia hoʻi hāʻawe, pōʻino i ka paakiki iwi papa.
  • Kūʻai ai 'wale nō ae keʻena kūʻai lāʻau lapaʻau.
  • I ka loaa ana i ka luna-i oleloia pae o ka lapaau mau ma ka lā, a ma bedtime e ana ai i ke koko,.
  • Lawe ka lapaʻauʻia no ka kiʻekiʻe ke koko, i hāpai keiki, eʻoiaʻiʻo, e pili ana me ke kauka.

He nui no ka maopopo i ka overdose o kēia mau ai 'ke alakai i ka undesirable hopena.

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