Ola kino, Hoomakaukau
Product "Levodopa": aʻo no ka hoʻohana 'ana, hōʻikeʻano, haku mele' ana, analogs a me nā hōʻike manaʻo
He aha mea i ka lāʻau "Levodopa"? Na Ke Kumu no ka hoʻohana, kūʻai, e e kūkākūkā i iki ae hōʻike manaʻo e pili ana i ka waiʻona. Oe e hoi aʻo e pili ana i ka mea i hoakaka ia keia ka lapaʻauʻia, ina loaa ia ia kekahi adverse reactions a me contraindications, ma i hana ia mea i loaʻa no ka kuai, i ka mea i komo i loko o kona haku mele 'ana, a no laila, ma luna o.
I ka haku mele 'ana, kinona, hōʻikeʻano
A eiiiiiaiou kekahi i ka lāʻau "Levodopa"? Na Ke Kumu no ka hoʻohana i ka 'ia ka hana' Oponopono o ka lāʻau mea levodopa. Ma ke kuai ana ia mea i loko o ka palapala o ka hoʻopoepoe spigot papa keʻokeʻoʻeleʻele, pūʻolo helu ma ka contour aeea a me ka pepa pahu, niioaaonoaaiii.
I ka rula o ka hana ana o ka medicament
lāʻau "Levodopa" Pehea 'aʻole ia hana? Na Ke Kumu no ka hoʻohana 'ana, ua hōʻike hōʻike manaʻo i kēia me ka hui pu antiparkinsonian Agena. Ua AIM e hoʻopau i ka rigidity, hypokinesia, tremor, drooling a me ka dysphagia.
Ma ke kino, e hana ka lapaʻauʻia ke keʻena ua hoohuliia i ka dopamine (CNS), hiki ana i ka shortage o ka hehee ai.
Dopamine e ia lŘlŘ iʻike ākea nā'aʻaʻa, hōʻike i Anati-Parkinson hopena o ka levodopa. O ke kumu ho i ka mea i ka mea, aole i komo iloko o ka Central ko mākou hopohopo'ōnaehana a me ka mea i ka kumu nui o adverse reactions o ka lāʻau.
E emi i ka mahele lāʻau o ka mea hana waiwai i loko o ke kanaka kino ua häʻawi mai medicament ma ka hoʻohui pū 'ia me nā mea kūpaleʻike ākea dopa-decarboxylase. Kēiaʻano hana kōkua, e emi ma kaʻaoʻao ona mai ka lawe i ka huaale.
Pharmacokinetics
Pehea ka nui o ka lapaʻauʻia ka paka "Levodopa"? Na Ke Kumu ma ka noi Huipuia, i ma hope o noho ai ka lāʻau i loko o ke kino ka mea, ua hala loa hoʻomaka koke ke kemu, mai ka liʻiliʻi.
Omo o kaʻeleu waiwai mea ma kahi o 20-30%. Ma keia pākōlea ia i malamaia ma hope ma kahi o 3 h.
Foodʻai ana (a me kekahi mauʻai) pono e loli ai i ka omo o ka lāʻau.
Ka lāʻau 'Ua metabolized, ma ia ho okumu i kekahi mau metabolites. Excretion o kaʻeleu waiwai i wahi ma nā puʻupaʻa, a ma ka naʻau liʻiliʻi.
nāʻikepili
Ma lalo o ka rula e hoomanawanui i hoakaka o ka lāʻau "Levodopa"? Na Ke Kumu no ka hoʻohana e like me ka hahai ana i nāʻikepili:
- postencephalitic maʻi pale e ia lŘlŘ ma cerebrovascular maʻi aʻawahia intoxication;
- Parkinson ka maʻi pale, eia hoi, i i ke kumu ma ka hoʻohana 'ana i antipsychotic ai';
- Parkinson ka maʻi.
Contraindications
Ina he mau contraindications ma "L-dopa" ia waiʻona? Na Ke Kumu no ka hoʻohana mau moʻolelo i kēia ka lapaʻauʻia ua papaia e lawe i ka i kēia hihia.
- hypersensitivity i na eiiiiiaiou;
- hui me Mao nā mea kūpale;
- i hāpai keiki, a i ka umauma-e hanai ana oia i kekahi kamaiki;
- hoʻomanawanui iki mai ma lalo o makahiki 18.
Me ka malama nui i ka lāʻau hiki ke hoonohoia ma:
- emphysema;
- imua o ke akemāmā maʻi, naau maʻi, ake a me ka endocrine'ōnaehana a me ka wahi;
- bronchial asthma;
- hoike ana mai o ka psychosis;
- melanoma (me mōʻaukala);
- huina-panina glaucoma;
- repetitive kāʻili 'ana (convulsions);
- hamama-huina glaucoma, a ia lŘlŘ i loko o ka maʻi palapala;
- hakuʻala, a ake ole;
- myocardial infarction (mōʻaukala), a me ka ano o ka acee? iuo oeiia o arrhythmias no hoi;
- duodenal ulcer a me ka'ōpū;
- CNS hoikeana o ka hookaumaha;
- naau pāpana ka haunaele.
Ka lāʻau 'o "L-dopa": kauoha no ka hoʻohana
Description o ka lāʻau i ua hōʻike mai iā ia ma luna. E like me ka mea, e ia?
E like me na kuhikuhi, ka lāʻau ua lawe hōʻike waha. Ka laʻau heluna Ua kiʻekiʻe o māhuahua aʻe mai ka palena iki a hiki i ka i kā mākou (ke kaumaha ma muli o ka kanaka hoʻomanawanui).
Ka hoʻomaka 'lapaʻau me ka mahele lāʻau o 0.25-1 g. Kēia huina Ua maheleia i ekolu apana. Ka laʻau heluna ua i nā mahuahua i 0,125-0,75 g. E hanaʻoe i ka mea i like manawa o ka manawa (e laʻa me,ʻekolu lā), hoʻomālama ma ke kanaka ahonui i ka pane, i hiki i ka manawa i ka wa a na kaʻoi loa ia e e malama mai i ka Inc.
ʻO kā mākou mahele lāʻau no ka lā e ole mamua o ewalu nā huna.
Ka lapaʻauʻia i loko o kekahi hihia, e mai ana ia. Ua oki ka lawe ia i nā.
Adverse reactions
I kaʻaoʻao 'ole o ka lāʻau "Levodopa"? Na Ke Kumu no ka ho ohana i hākālia nō ia i loko o ka pōʻaiapili o kona? Eaia i ke kanaka i 'ike i kekahi adverse reactions i aloha ia i ka hana o nā nenoai o ke kino.
- Mea'ōnaehana mānowai koko'ōnaehana: naau palpitations, arrhythmia, haunaele o ka puʻe, orthostatic reactions, syncope, a no laila, ma luna o.
- Digestive'āpana: diarrhea, ka luaʻi, dyspepsia, anorexia, constipation, loli ma ka ho'āʻoʻana, maloo waha, kahe ana ke koko mai ka gastrointestinal'āpana.
Ua E hoi e kaulana i ole hoʻokoe 'ʻaoʻao reactions mea e pono ai ka hana o ka hematopoiesis, urinary, naehana hanu, a me ko mākou hopohopo nenoai. Pinepine i loko o nā mea maʻi e loaa ana keia k allergic reactions ana, loli ma ka keʻena hoʻokolohua kiko'î a undesirable 'ole ma luna o kaʻili.
Hihia o ka overdose (symptoms, lapaʻau)
I ana kiʻekiʻe nā māhele hōʻike he nui holomua o kaʻaoʻao loa. Mau kumu koi lapaau i loko o ka palapala o ka lavage, ke hoʻomanawanui i ka nui ana ka mālamaʻana a me ka hana ana o ka naau. Inā pono, e lawe mai antiarrhythmic Inc.
lāʻau hana kūleʻa
I ka wā hoʻokahi? Eaia a me ka noonoo ana o ka la hoomalolo "ditilina" Hoʻokolohua-agonists, a me ka konohiki mea i manao ia no ka inhalation anesthesia, maoli ka likelihood o arrhythmias o ka naau.
Bioavailability "Levodopa" ke emi i ka tricyclic antidepressants.
I ka hoʻohuiʻia o ka lāʻau a me "thioxanthenes," "Diazepam" antipsychotic "Phenytoin" ka m-holinoblokatorami "clonidine", "Difenilbutilpiperidinom" "Papaverine", "Clozapine", "phenothiazine" "pyridoxine" a me ka "reserpine" muli o kona kulana pinepine ia ho'ēmi i kā kona antiparkinsonian ai.
Likiuma mea haʻilula keimikala hoomahuahua i ka pahiki o ka hanana o dyskinesias a me hallucinations, a "methyldopa" medicament maoli heʻaoʻao reactions.
Ka hui malu pu ana o Mao nā mea kūpale , a "Levodopa" hiki aku i ka hoʻopōʻino holo. Ma keia manao, e ka wā mawaena ma waena o nā māhele o kēia mau lapaʻauʻia pono ma ka liʻiliʻi 14 lā.
Na hiohiona ka ho'ēmiʻana i loko o ka puʻuwai malama me ka huihui 'ana o ka lapaʻauʻia a me ka noonoo "tubocurarine".
Uluwehi O "metoclopramide" e māhuahua bioavailability "Levodopa" accelerating gastric emptying. Kēia ke kūlana maikaʻiʻole i ka papa o ka mea maʻi.
I Kekahi Mau koi no ka hoʻohana ana i ka lāʻau '
He aha kou pono e ike mua e lawe i ka papa "Levodopa"? Na Ke Kumu no ka hoʻohana (ke kumukuai ma lalo nei), noka mea e pili ana i ka make māinoino e ola ma abrupt ke kāpaeʻana o ka medicament.
Ma na wahi he mea hiki ole ke pale ia i ka ka ho'ēmiʻana o ka laʻau heluna paha withdrawal o ka lapaʻauʻia noi aku maʻamau ka mālamaʻana o ka hoʻomanawanui ka kulana.
Ma mua o ka lāʻau 'aʻole pono e hoʻopauʻai waiwai ma ka kumuʻiʻo, no ka mea, ho'ēmi i kā ka absorbability o kaʻeleu waiwai.
Ke Inc pono ana ka mālamaʻana o ka mea likeʻole nenoai, nā loko, a me nā mea kiko'î koko.
Price a me analogues
Ka hoʻopuniʻana analogues "L-dopa" hoomalolo 'o ia hoʻi mea e like me he "levodopa benserazide" a me ka "Levodopa Carbidopa". Na Ke Kumu no ka hoʻohana mau moʻolelo i kēia mau ai 'i ka ia nāʻikepili,ʻaoʻao' ole, maomeka o ka hana a me ka contraindications. Ka mea wale nō likeʻole ma waena o kēia mau kālā o lākou haku mele 'ana.
Ia hana 'ona e like me carbidopa a me benserazide emi i ka? Iecaianoaaiiie o dopamine iʻike ākea'aʻaʻa, hiki mahuahua i ka nui o ka levodopa komo i ka CNS.
Penei, ka mea hiki ke pakele ke kaulana i kuhikuhi "Levodopa Carbidopa" a me ka "levodopa benserazide" (kauoha no ka hoʻohana ana i kēia mau mea i kekahi i loko iho i loko o ka'ōpala) eliminates hou? Eaia nā mea kūpaleʻike ākea dopa-decarboxylase.
Like no ka mea'ē aʻe na¯, laila, i ka hope nā mea ai 'like "Isik Meath", "Tremonorm", "Dopar 275", "Tidomet", "Duellin', 'Sinemet', 'Zimoks", "Sindopa", "Isik" "Lake". Lakou pono koho wale kauka.
Ke kumukuai o ka "Levodopa" ka lāʻau Ua kiʻekiʻe. Ma keʻena kūʻai lāʻau lapaʻau, e hiki ke kuai i kēia ka lapaʻauʻia i loko o 1500-1850 rubles.
ka lapaʻauʻia Reviews
Lapaau ana i kekahi maʻi e halihaliia oia iwaho wale no ka mea o ka hoao ana i ka kauka. A me Parkinson ka mea i koe.
E hoomanawanui i ka poe i ka lāʻau "Levodopa" i loko o kona poli manao ana, aʻaʻole i ka maikaʻi pākōlea hopena. No laila, pinepine keia medicament hōʻike manaʻo i io. Mea hoʻohana i hoike ia e like me ka hooloihi ae i hoʻohana o ka lapaʻauʻia pepeiaohao nui hou i malama pono.
Inā ua laweʻia ka lapaʻauʻia ma lalo o noonoo ma ka noaia, i? Ac? Ma ka hoao ana i ka 'oihana e hahai i ka papa o ka maʻi, i ka iapaau ana kaʻina mea aneane manawa holomua. O ke kumu ho i ka mea e pono e lawe i kaʻeleu lāʻau i loko o ka ikaika laʻau heluna, i hilinaʻi nui ma ka hoomanawanui, me nā 'ano o ka maʻi a me ka' ē aʻe aʻe.
Nā mea maʻi i ikaika hooko ana me ka iapaau ana regimen, ua hai mai la ia i ka lāʻau "Levodopa" ka loa mana ma ka ola pilikia ke kāpaeʻana.
I ka mea, he nui ohumu e pili ana i ke kiʻekiʻe lilo o ka lapaʻauʻia. Eia naʻe, poe akamai i koi ia i ke kumu kuai o keia k ka pau hoaponoia.
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